2. Signaling Pathways
  3. Metabolic Enzyme/Protease
  4. Drug Metabolite

Drug Metabolite

Drug Metabolite

Related Products

PDF 3.95 MB

Drug metabolite results when a drug is metabolized into a modified form which continues to produce effects. Drug metabolism redox reactions such as heteroatom dealkylations, hydroxylations, heteroatom oxygenations, reductions, and dehydrogenations can yield active metabolites, and in rare cases even conjugation reactions can yield an active metabolite.

Cat. No. Product Name Effect Purity Chemical Structure
  • HY-W072459A
    6'-Hydroxydihydrocinchonidine acetate
    6'-Hydroxydihydrocinchonidine acetate is a metabolite of Quinine (HY-D0143) (antimalarial agent).
    6'-Hydroxydihydrocinchonidine acetate
  • HY-W144077
    Permethric acid
    Permethric acid is a metabolite of insecticide permethrin.
    Permethric acid
  • HY-133672
    (Rac)-Mono(3,5,5-trimethylhexyl) phthalate
    (Rac)-Mono(3,5,5-trimethylhexyl) phthalate is a important metabolite of commonly used phthalate plasticizers. (Rac)-Mono(3,5,5-trimethylhexyl) phthalate has immuno-suppressive effect.
    (Rac)-Mono(3,5,5-trimethylhexyl) phthalate
  • HY-W775325
    7-Hydroxycannabidiol
    7-Hydroxycannabidiol (7-OH-CBD) is the metabolite of cannabidiol, which could be found in human serum and saliva.
    7-Hydroxycannabidiol
  • HY-116787R
    5-Hydroxythiabendazole (Standard)
    5-Hydroxythiabendazole (Standard) is the analytical standard of 5-Hydroxythiabendazole. This product is intended for research and analytical applications. 5-Hydroxythiabendazole (5-OHTBZ) is a biomarker of Thiabendazole (HY-B0263) exposure.
    5-Hydroxythiabendazole (Standard)
  • HY-13256AS
    Desmethyl Erlotinib-d4
    Desmethyl Erlotinib-d4 is the deuterium labeled Desmethyl Erlotinib. Desmethyl Erlotinib (OSI-420 free base) is an active metabolite of Erlotinib. Erlotinib is a potent EGFR tyrosin kinase inhibitor. Desmethyl Erlotinib-d4 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
    Desmethyl Erlotinib-d<sub>4</sub>
  • HY-Z7429
    3-Hydroxy-4-methyl-2(5H)-thiophenone
    3-Hydroxy-4-methyl-2(5H)-thiophenone (compound 18) is a pyrazine derivative and the major acidic degradation product of Cephalexin (HY-B0200).
    3-Hydroxy-4-methyl-2(5H)-thiophenone
  • HY-172055
    PB-22 N-(5-Hydroxypentyl)-3-carboxyindole metabolite
    PB-22 N-(5-Hydroxypentyl)-3-carboxyindole metabolite is a metabolite of PB-22. PB-22 is a cannabinoid.
    PB-22 N-(5-Hydroxypentyl)-3-carboxyindole metabolite
  • HY-145482R
    W36017 (Standard)
    8-Hydroxyquinoline (hemisulfate) (Standard) is the analytical standard of 8-Hydroxyquinoline (hemisulfate). This product is intended for research and analytical applications. 8-Hydroxyquinoline hemisulfate (8-Quinolinol hemisulfate) is a monoprotic bidentate chelating agent, exhibits antiseptic, disinfectant, and pesticide properties, functioning as a transcription inhibitor.
    W36017 (Standard)
  • HY-W002065R
    4-Carboxypyrazole (Standard)
    4-Carboxypyrazole is an endogenous metabolite.
    4-Carboxypyrazole (Standard)
  • HY-W714541
    N-Acetyl-S-(2-cyanoethyl)-L-cysteine ammonium
    N-Acetyl-S-(2-cyanoethyl) -L-cysteine ammonium salt is the urinary metabolite of acrylamide in vivo.
    N-Acetyl-S-(2-cyanoethyl)-L-cysteine ammonium
  • HY-139232
    17(R)-Resolvin D3
    17(R)-Resolvin D3 is a metabolite of docosahexaenoic acid (DHA). 17(R)-Resolvin D3 has anti-inflammatory activity.
    17(R)-Resolvin D3
  • HY-W740165
    Desmethyl Levofloxacin hydrochloride
    Desmethyl Levofloxacin hydrochloride is an antibacterial agent with broad-spectrum antibacterial activity against a variety of pathogens. Desmethyl Levofloxacin hydrochloride effectively fights bacterial infections by inhibiting bacterial DNA synthesis. Studies on Desmethyl Levofloxacin hydrochloride have shown that it has potential in inhibiting respiratory infections.
    Desmethyl Levofloxacin hydrochloride
  • HY-166341S
    S 8849-1-d4 free base
    S 8849-1-d4 (free base) (Tianeptine metabolite MC5-d4) is deuterium labeled S 8849-1 (free base). S 8849-1 (free base) (Tianeptine metabolite MC5) is a Tianeptine (HY-90003) metabolite that is found in plasma. The mean elimination half-lives of S 8849-1 (free base) is 7.53 h in rats. S 8849-1 (free base) is promising for research of antidepressants.
    S 8849-1-d<sub>4</sub> free base
  • HY-W338799
    Disulfoton sulfone
    Disulfoton sulfone is a metabolite of the organophosphorus pesticide Disulfoton.
    Disulfoton sulfone
  • HY-Z6663
    Salbutamol methyl ether
    Salbutamol methyl ether is a derivative of Salbutamol (HY-B1037) used as an immunohapten to obtain antibodies.
    Salbutamol methyl ether
  • HY-I0169R
    (R)-Amino-N-benzyl-3-methoxypropionamide (Standard)
    (R)-Amino-N-benzyl-3-methoxypropionamide (Standard) is the analytical standard of (R)-Amino-N-benzyl-3-methoxypropionamide. This product is intended for research and analytical applications. (R)-Amino-N-benzyl-3-methoxypropionamide is a stable intermediate of Lacosamide (an antiepileptic drug).
    (R)-Amino-N-benzyl-3-methoxypropionamide (Standard)
  • HY-137238
    Ethyl mycophenolate
    Ethyl mycophenolate is a potential impurity found in commercial preparations of the mycophenolic acid prodrug mycophenolate mofetil.
    Ethyl mycophenolate
  • HY-N8500
    Aristolochic acid Ia
    Aristolochic acid Ia is an oxidative metabolite of aristolochic acid I, which can be used to study the detoxification pathway of aristolochic acid metabolism.
    Aristolochic acid Ia
  • HY-W436495
    6,15-Diketo-13,14-dihydro prostaglandin F1α
    6,15-Diketo-13,14-dihydro prostaglandin F1α (6,15-Diketo-13,14-dihydro-PGF1α) is a metabolite of prostacyclin (PGI2). 6,15-Diketo-13,14-dihydro prostaglandin F1α enhances intracellular cAMP and cholesterol metabolism in bovine arterial smooth muscle cells.
    6,15-Diketo-13,14-dihydro prostaglandin F1α
Cat. No. Product Name / Synonyms Application Reactivity